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Prostate cancer–associated SPOP mutations confer resistance to BET inhibitors through stabilization of BRD4

  • Xiangpeng Dai
  • , Wenjian Gan
  • , Xiaoning Li
  • , Shangqian Wang
  • , Wei Zhang
  • , Ling Huang
  • , Shengwu Liu
  • , Qing Zhong
  • , Jianping Guo
  • , Jinfang Zhang
  • , Ting Chen
  • , Kouhei Shimizu
  • , Francisco Beca
  • , Mirjam Blattner
  • , Divya Vasudevan
  • , Dennis L Buckley
  • , Jun Qi
  • , Lorenz Buser
  • , Pengda Liu
  • , Hiroyuki Inuzuka
  • , Andrew H Beck
  • , Liewei Wang
  • , Peter J Wild
  • , Levi A Garraway
  • , Mark A Rubin
  • , Christopher E Barbieri
  • , Kwok-Kin Wong
  • , Senthil K Muthuswamy
  • , Jiaoti Huang
  • , Yu Chen
  • , James E Bradner
  • , Wenyi Wei

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